Umbralisib R-enantiomer (RP5264 R-enantiomer) is a delta inhibitor of PI3K and a less active enantiomer of TGR-1202. The IC50 of Umbralisib R-enantiomers against deltaPI3 kinase is at least 20 times lower than that of the inhibitors against other PI3K isoforms (A, beta, and gamma).
Molecular Weight:
571.55
Purity:
95.61%
CAS Number:
[1532533-69-9]
Formula:
C31H24F3N5O3
Target:
PI3K
T13140
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