BMS-986158 is a highly effective BET inhibitor, demonstrating IC50 values of 6.6 nM in NCI-H211 small cell lung cancer (SCLC) cells and 5 nM in MDA-MB231 triple negative breast cancer (TNBC) cells.
Molecular Weight:
495.62
Purity:
98.78%
CAS Number:
[1800340-40-2]
Formula:
C30H33N5O2
Target:
Epigenetic Reader Domain
T14685
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