CAY10566 shows excellent cellular activity in blocking the conversion of saturated long-chain fatty acid-CoAs (LCFA-CoAs) to monounsaturated LCFA-CoAs in HepG2 cells (IC50=7.9 nM or 6.8 nM). CAY10566 is a potent, orally bioavailable and selective stearoyl-CoA desaturase1 (SCD1) inhibitor with IC50s of 4.5 and 26 nM in mouse and human enzymatic assays, respectively..
Molecular Weight:
389.81
Purity:
99.50%
CAS Number:
[944808-88-2]
Formula:
C18H17ClFN5O2
Target:
Dehydrogenase|||Stearoyl-CoA Desaturase (SCD)
T14878
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