CMPD101 is a membrane-permeable small-molecule inhibitor of GRK2/3 (IC50: 18 nM and 5.4 nM). Which can be used for the study of heart failure. CMPD101 exhibits less selectively against GRK1, GRK5, ROCK-2 and PKCalpha with IC50s of 3.1 µM , 2.3 µM, 1.4 µM and 8.1 µM, respectively.
Molecular Weight:
466.46
Purity:
98.34%
CAS Number:
[865608-11-3]
Formula:
C24H21F3N6O
Target:
ROCK|||GRK|||PKC
T14989
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