KDM5A-IN-1 is an orally available, potent and selective inhibitor of the pan-histidine lysine demethylase 5 KDM5, inhibiting KDM5A, KDM5B, and KDM5C with IC50 values of 45 nM, 56 nM, and 55 nM, respectively.KDM5A-IN-1 inhibits PC9 H3K4Me3, and may be useful in cancer research.
Molecular Weight:
290.36
Purity:
>99.99%
CAS Number:
[1905481-36-8]
Formula:
C15H22N4O2
Target:
Histone Demethylase
T15650
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