Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83) that blocks recall in fear conditioning in mice. It exhibits inverse agonist and antagonist activity (Ki, 220 nM) at the A2A receptor and weak antagonist activity (Ki, 736 nM) at the 5-HT2B receptor.
Molecular Weight:
307.35
Purity:
99.50%
CAS Number:
[1309198-71-7]
Formula:
C17H17N5O
Target:
Adenosine Receptor|||GPCR|||5-HT Receptor
T16378
* VAT and and shipping costs not included. Errors and price changes excepted
