PF-04995274, CAS [[1331782-27-4]]

Catalog Number: TGM-T16481
Article Name: PF-04995274, CAS [[1331782-27-4]]
Biozol Catalog Number: TGM-T16481
Supplier Catalog Number: T16481
Alternative Catalog Number: TGM-T16481-1MLX10MM(INDMSO),TGM-T16481-1MG,TGM-T16481-5MG,TGM-T16481-10MG,TGM-T16481-25MG,TGM-T16481-50MG,TGM-T16481-100MG
Manufacturer: TargetMol
Category: Biochemikalien
PF-04995274 is an effective, high-affinity, and partial serotonin 4 receptor (5-HT4R) agonist. PF-04995274 is brain penetrant and can be used for cognitive disorders associated with Alzheimers disease. PF-04995274 has an EC50 range of 0.26-0.47 nM for human 5-HT4A/4B/4D/4E (Ki range of 0.15-0.46 nM). It also has an EC50 range of 0.59-0.65 nM for rat 5-HT4S/4L/4E (Ki of 0.30 nM for rat 5-HT4S).
Molecular Weight: 432.51
Purity: 99.52%
CAS Number: [1331782-27-4]
Formula: C23H32N2O6
Target: 5-HT Receptor
T16481