Pozanicline hydrochloride is an orally bioavailable nicotinic acetylcholine receptor (nAChR) agonist with a Ki of 16.7 nM for binding to [3H]cytisine sites[1]. Pozanicline hydrochloride is an alpha4beta2-selective nAChR agonist, which binds to rat brain alpha4beta2 nAChR with a Ki of 17 nM while binding to alpha7 nAChR is insignificant[2].
Molecular Weight:
228.72
Purity:
97.13%
Formula:
C11H17ClN2O
Target:
AChR
T16563L
* VAT and and shipping costs not included. Errors and price changes excepted