GSK-5959 is an effective, specific and cell permeable BRPF1 bromodomain inhibitor (IC50: ~80 nM). The selectivity of GSK-5959 for BRPF1 is >100-fold over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains.
Molecular Weight:
394.47
Purity:
98.35%
CAS Number:
[901245-65-6]
Formula:
C22H26N4O3
Target:
Epigenetic Reader Domain
T1972
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