SR-12062 functions as a full agonist at neurotensin receptor 1 (NTSR1), demonstrating notable efficacy and increased potency. Its EC50 value on NTSR1 is 2 µM, with complete receptor activation (Emax=100%). Compared to the parent compound 1 (EC50=178 µM, Emax=17%), SR-12062 shows approximately 90-fold greater potency.
Molecular Weight:
415.48
CAS Number:
[1623019-77-1]
Formula:
C25H25N3O3
T202825
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