Fluorphine, an analog of Brorphine, binds to the µ-opioid receptor (MOR) with a Ki of 12.5 nM. It exhibits GTPgammaS binding activity with an EC50 of 75 nM and beta-arrestin 2 recruitment activity with an EC50 of 377 nM, and it also has respiratory depressive effects.
Molecular Weight:
339.41
CAS Number:
[6440-42-2]
Formula:
C20H22FN3O
Target:
Opioid Receptor
T203493
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