PKN3-IN-1 (compound 16) inhibits PKN3 (serine/threonine-protein kinase N3) and GAK (cyclin G-associated kinase) with an IC50 of 0.014 µM and a Ki of 0.0044 µM. PKN3-IN-1 is a potential tool compound for investigating the cell biology of PKN3 and its role in pancreatic and prostate cancers, as well as T-cell acute lymphoblastic leukemia.
Molecular Weight:
436.244
CAS Number:
[2361545-75-5]
Formula:
C18H17IN2O3
Target:
PI3K
T204631
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