GABAA receptor modulator-4 (Compound 4) acts as a negative allosteric modulator of the GABAA receptor. It inhibits the peak and steady-state currents mediated by the alpha1beta3gamma2 GABAA receptors, with an IC50 of 10 µM for both.
Molecular Weight:
373.26
Formula:
C15H17BrO4S
Target:
GABA Receptor
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