EN1441 is a covalent degrader that targets the androgen receptor (AR) with an EC50 value of 4.2 µM, as well as its truncated variant AR-V7. It selectively and effectively degrades AR and AR-V7 in androgen-independent prostate cancer cells. EN1441 holds potential for research into androgen-independent prostate cancer.
Molecular Weight:
264.708
CAS Number:
[2196448-47-0]
Formula:
C13H13ClN2O2
Target:
Androgen Receptor
T206982
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