PIPE-3297 (compound 25) is a selective kappa opioid receptor (KOR) agonist that activates the G protein signaling pathway with an EC50 of 1.1 nM and exhibits low beta-arrestin-2 recruitment activity (10%). Additionally, PIPE-3297 promotes myelination and has anti-inflammatory properties.
Formula:
C23H30N2O
Target:
Opioid Receptor
* VAT and and shipping costs not included. Errors and price changes excepted
