Keap1-Nrf2-IN-19 (compound 33) is an orally active inhibitor of the Keap1-Nrf2 protein-protein interaction (PPI), with a Kd value of 0.0014 µM. Keap1-Nrf2-IN-19 exhibits less than 50% inhibition of hERG at 30 µM and CYPs at 10 µM.
Formula:
C25H27FN2O4
Target:
Nrf2
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