VU6008055 is a potent, selective, orally bioavailable M4 positive allosteric modulator that can cross the blood-brain barrier. It exhibits EC50 values of 73.4 nM for hM4 and 19.5 nM for rM4, and it demonstrates antipsychotic-like activity.
Molecular Weight:
379.48
CAS Number:
[2170551-59-2]
Formula:
C20H21N5OS
Target:
AChR
T210756
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