RS-79948-197 hemihydrate is a non-imidazoline alpha2-adrenoceptor antagonist. It exhibits Kd values of 0.42 nM, 0.18 nM, and 0.19 nM for rat alpha2A, alpha2B, and alpha2C receptors, respectively, and 0.60 nM, 0.46 nM, and 0.77 nM for human alpha2A, alpha2B, and alpha2C receptors.
Target:
Adrenergic Receptor
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