BI-9466 (Compound 2) is an antagonist of the NSD3-PWWP1 domain with a dissociation constant (Kd) of 144 µM. Designed as a negative control compound for BI-9321, BI-9466 lacks inhibitory activity against the NSD3-PWWP1 domain due to a more basic azacyclic structure introduced at the 5-position of BI-9321.
Molecular Weight:
295.38
CAS Number:
[2538293-52-4]
Formula:
C17H21N5
Target:
Histone Methyltransferase
T212115
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