Azepexole dihydrochloride (B-HT 933), a potent and selective alpha 2-adrenoceptor agonist, exhibits affinity for alpha2A-, alpha2B-, and alpha2C-adrenoceptor subtypes with pKis of 8.3, 7.6, and 7.5, respectively [1]. It elicits a concentration-dependent inhibition of peristaltic contractions, evidenced by an IC50 of 78.72 nM.
Molecular Weight:
254.16
CAS Number:
[36067-72-8]
Formula:
C9H17Cl2N3O
Target:
Others|||Adrenergic Receptor
T21787
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