()-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM). J-113397 inhibited nociceptin/orphanin FQ-stimulated GTPgammaS binding to CHO cells expressing ORL1 with an IC50 value of 5.3 nM. J-113397 can be used for researching the physiological roles of nociceptin/orphanin FQ [1].
Molecular Weight:
399.57
CAS Number:
[217461-40-0]
Formula:
C24H37N3O2
Target:
Others|||Opioid Receptor
T21999
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