AMI-1 free acid is a potent, cell-permeable, and reversible inhibitor of protein arginine N-methyltransferases (PRMTs), with inhibitory concentration 50 (IC50) values of 8.8 µM for human PRMT1 and 3.0 µM for yeast-Hmt1p. It achieves its PRMTs inhibitory activity by obstructing peptide-substrate binding [1].
Molecular Weight:
504.49
Purity:
97.80%
CAS Number:
[134-47-4]
Formula:
C21H16N2O9S2
Target:
Histone Methyltransferase
T22239
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