CP-100356 hydrochloride is an orally active, low micromolar dual inhibitor of MDR1 (P-gp) and BCRP, a nucleotide-derived substrate analogue that inhibits MDR1-mediated Calcein-AM and BCRP-mediated Prazosin transporters. Additionally, CP-100356 inhibits OATP1B1 and induces stomatal opening in the dark.
Molecular Weight:
597.1
Purity:
99.19%
CAS Number:
[142715-48-8]
Formula:
C31H37ClN4O6
Target:
P-gp|||BCRP
T22680
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