SR1664 is a potent and selective PPARgamma inhibitor with potential antidiabetic activity. SR1664 binds to PPARgamma and potently inhibits Cdk5-mediated PPARgamma phosphorylation (IC50 = 80 nM, Ki = 28.67 nM) without exhibiting PPARgamma agonist activity.
Molecular Weight:
547.6
Purity:
99.43%
CAS Number:
[1338259-05-4]
Formula:
C33H29N3O5
Target:
PPAR
T23389
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