FT001 is a potent, selective and orally available inhibitor of BET Bromodomain with antitumor activity. FT001 inhibited the expression of MYC with the IC50 value of 0.46 µM). FT001 has potent antiproliferative effects against MV-4-11 and demonstrates significant MYC mRNA suppression both in vitro and in vivo.
Molecular Weight:
467.58
Purity:
>99.99%
CAS Number:
[1778655-51-8]
Formula:
C25H29N3O4S
Target:
Epigenetic Reader Domain
T27392
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