SKI2496 is a potent and orally bioavailableantagonist of Gonadotropin-Releasing Hormone Receptor (hGnRHR IC50 = 0.46 nM, max. LH inh. inh. (%, h)= 84%, 12h, LH inh. (24h) = 76%.). SKI2496 exhibits more selective antagonistic activity toward the human GnRH receptors over the GnRHRs in monkeys and rats.
Molecular Weight:
739.68
CAS Number:
[1308378-95-1]
Formula:
C35H36F7N5O5
Target:
ERK|||Others|||GNRH Receptor
T28795
* VAT and and shipping costs not included. Errors and price changes excepted