MTI-31 (LXI-15029) is a potent, orally active, and highly selective inhibitor of mTORC1 and mTORC2, exhibiting a Kd of 0.20 nM for mTOR and >5,000-fold selectivity over PIK3CA, PIK3CB, and PIK3G in binding assays, with an IC50 of 39 nM for mTOR in a LANCE assay of mTOR substrate phosphorylation with 100 µM ATP [1].
Molecular Weight:
474.55
Purity:
99.76%
CAS Number:
[1567915-38-1]
Formula:
C26H30N6O3
Target:
mTOR
T35343
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