P38alpha Inhibitor 2, a potent and selective inhibitor of p38alpha MAPK, exhibits a pIC50 value of 9.6. It also demonstrates inhibition of the hERG ion channel (IC50=27 µM) and maintains promising selectivity, with <30% inhibition across a panel of 51 protein kinases at a 10 µM concentration and a broad specificity against 141 other biological targets[1].
Molecular Weight:
475.58
CAS Number:
[1095003-80-7]
Formula:
C27H33N5O3
Target:
Others|||p38 MAPK
T36012
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