GABAA receptor antagonist that binds the picrotoxin site and stabilizes the inactive form of the channel via allosteric interaction. Accelerates the decay of GABA-induced Cl- currents with little effect on peak amplitude. Also inhibits 5-HT3A receptors via a similar mechanism.
Molecular Weight:
299.37
Purity:
99.65%
CAS Number:
[152273-12-6]
Formula:
C17H21N3O2
Target:
GABA Receptor
T3644
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