Rolapitant (SCH619734) hydrochloride is a potent, selective, long-acting, and orally active neurokinin 1 (NK1) receptor antagonist with a K_i of 0.66 nM, which does not interact with CYP3A4 and demonstrates potent centrally-mediated anti-emetic activity in both acute and delayed ferret emesis models [1] [2].
Molecular Weight:
536.94
Purity:
99.79%
CAS Number:
[858102-79-1]
Formula:
C25H27ClF6N2O2
Target:
Neurokinin receptor
T3724
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