Desmethyl bosentan, an active metabolite of the endothelin receptor antagonist bosentan, activates the pregnane X receptor (PXR) in CV-1 monkey kidney cells expressing the human receptor in a reporter assay at a concentration of 25 µM.
Molecular Weight:
537.59
CAS Number:
[253688-61-8]
Formula:
C26H27N5O6S
Target:
Drug Metabolite|||Others|||Cytochromes P450
T37351
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