CAY10771 is a dual agonist of farnesoid X receptor (FXR) and peroxisome proliferator-activated receptor delta (PPARdelta).1It activates FXR and PPARdelta in reporter assays using HEK293T cells (EC50s = 0.94 and 1.5 µM, respectively) and is selective for these receptors over retinoic acid receptor alpha (RARalpha), retinoid X receptor alpha (RXRalpha), PPARalpha, PPARgamma, and liver X receptor alpha (LXRalpha) at 10 µM.
Molecular Weight:
559.87
CAS Number:
[2522599-79-5]
Formula:
C28H25Cl3N2O4
Target:
Others
T37414
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