Dapolsertib (SEL24-B489) is an orally bioavailable and potent PIM and FLT3-ITD inhibitor, inhibiting PIM1, PIM2, and PIM3, decreasing PIM substrate phosphorylation, and inducing dose-dependent apoptosis in leukemia cells.
Molecular Weight:
446.14
Purity:
99.61%
CAS Number:
[1616359-00-2]
Formula:
C15H18Br2N4O2
Target:
FLT|||Apoptosis|||Pim
T39085
T39085
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