KML29 is highly selective and effective monoacylglycerol lipase (MAGL) inhibitor. It has effective inhibition of human/mouse/rat MAGL (IC50: 5.9/15/43 nM). It has not inhibitory for FAAH (IC50 > 50 µM). It also effectively and selectively blocks hydrolysis of 2-arachidonoylglycerol (2-AG) in mice (IC50: 2.5 nM, 2-AG, >50 µM, AEA).
Molecular Weight:
549.42
Purity:
98.16%
CAS Number:
[1380424-42-9]
Formula:
C24H21F6NO7
Target:
Lipase|||MAGL
T4052
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