PBRM1-BD2-IN-8 (compound 34) is a potent PBRM1 Bromodomain inhibitor with PBRM1-BD2 Kd of 4.4 µM, PBRM1-BD2 IC50 of 0.16 µM, and PBRM1-BD5 Kd of 25 µM, PBRM1-BD2-IN-8 shows anti-cancer activity.
Molecular Weight:
317.18
Purity:
99.48%
CAS Number:
[2819989-75-6]
Formula:
C15H13BrN2O
Target:
Epigenetic Reader Domain
T60157
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