DYRK1-IN-1 is a highly selective and ligand-efficient DYRK1A inhibitor that inhibits DYRK1A phosphorylation activity with an IC50 value of 220 nM. It exhibits good permeability and cellular activity without P-glycoprotein liability, making it suitable for research on central nervous system penetrant DYRK1A chemical probes [1].
Molecular Weight:
240.26
CAS Number:
[2814486-79-6]
Formula:
C12H12N6
Target:
DYRK|||Others
T60334
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