KDM4-IN-4 (compound 47) is a potent inhibitor of histone lysine demethylase 4 (KDM4), with a binding constant of approximately 80 µM for the KDM4A-Tudor domain. It inhibits H3K4Me3 binding to the Tudor domain in cellular contexts with an EC50 value of 105 µM, holding potential for anticancer research applications [1].
Molecular Weight:
245.36
Purity:
0.9961
CAS Number:
[2230475-63-3]
Formula:
C16H23NO
Target:
Histone Demethylase
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