TAK-285, CAS [[871026-44-7]]

Catalog Number: TGM-T6039
Article Name: TAK-285, CAS [[871026-44-7]]
Biozol Catalog Number: TGM-T6039
Supplier Catalog Number: T6039
Alternative Catalog Number: TGM-T6039-1MLX10MM(INDMSO), TGM-T6039-1MG, TGM-T6039-5MG, TGM-T6039-10MG, TGM-T6039-25MG, TGM-T6039-50MG, TGM-T6039-100MG, TGM-T6039-200MG
Manufacturer: TargetMol
Category: Biochemikalien
Alternative Names: TAK285 , TAK 285
TAK-285 is a novel dual HER2 and EGFR(HER1) inhibitor with IC50 of 17 nM and 23 nM, >10-fold selectivity for HER1/2 than HER4, less potent to MEK1/5, c-Met, Aurora B, Lck, CSK etc. Phase 1.
Molecular Weight: 547.96
Purity: 0.9973
CAS Number: [871026-44-7]
Formula: C26H25ClF3N5O3
Target: MEK|||EGFR|||Aurora Kinase|||HER