Fenspiride is an antagonist of H1-histamine receptors. Fenspiride is an orally active non-steroidal anti-inflammatory agent that can be used for the treatment of respiratory tract infections and otitis media. Fenspiride inhibited phosphodiesterase 4 and phosphodiesterase 3 activities with -logIC50 values of 4.16+/-0.09 and 3.44+/-0.12, respectively. Phosphodiesterase 5 activity was also inhibited with a -logIC50 value of approximately 3.8.
Molecular Weight:
260.33
CAS Number:
[5053-06-5]
Formula:
C15H20N2O2
Target:
Others|||PDE|||Histamine Receptor
T60417
* VAT and and shipping costs not included. Errors and price changes excepted