Sapitinib (AZD-8931) , a reversible, ATP competitive inhibitor of EGFR(IC50=4 nM), ErbB2(IC50=3 nM) and ErbB3(IC50=4 nM), is more effective over Gefitinib or Lapatinib against NSCLC cell, 100-fold more specific for the ErbB family over MNK1 and Flt.
Molecular Weight:
473.93
Purity:
99.83%
CAS Number:
[848942-61-0]
Formula:
C23H25ClFN5O3
Target:
EGFR
T6092
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