IAA65 is a potent and highly selective transient receptor potential ankyrin 1 (TRPA1) inhibitor (IC50 = 4.3 nM). It demonstrates significant analgesic activity in animal models of inflammatory and neuropathic pain by competitively blocking TRPA1-mediated calcium influx in sensory neurons.
Molecular Weight:
365.27
CAS Number:
[2987139-96-6]
Formula:
C16H13F6NO2
Target:
TRP/TRPV Channel
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