20S Proteasome-IN-4 (Compound 7) is an orally active inhibitor of the 20S proteasome, selectively targeting the parasite form and demonstrating brain penetration capabilities. It exhibits a potent IC50 value of 6.3 nM against the T. b. brucei 20S proteasome, making it suitable for human African trypanosomiasis (HAT) research [1].
Molecular Weight:
421.83
CAS Number:
[2827061-47-0]
Formula:
C20H18ClF2N3O3
Target:
Others|||Parasite|||Proteasome
T62255
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