CCG-273220 is a covalent inhibitor of G protein-coupled receptor (GPCR) kinase 5 (GRK5) (IC50: 220 nM).CCG-273220 covalently binds the GRK5 subfamily-specific residue Cys474 and is more selective for GRK5 than GRK2.
Molecular Weight:
494.95
CAS Number:
[2750414-35-6]
Formula:
C26H24ClFN4O3
Target:
Others|||GRK
T63340
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