hA2A/hCA XII modulator 1 is a potent antagonist of the hA2A adenosine receptor (hA2AAR), a triazolopyrazine that acts on hA2AAR (Ki: 6.4 nM), hA1AR (Ki: 4.819 µM), and hA3AR (Ki>30 µM). hA2A/hCA XII modulator 1 Also a potent inhibitor of human carbonic anhydrase XII (hCA XII), capable of acting on hCA XII (Ki: 6.2 nM), hCA II (Ki: 46 nM), hCA IX (Ki: 466 nM) and hCA I (Ki: 8.351 µM). hA2A/hCA XII modulator 1 exhibits potential for cancer research.
Molecular Weight:
501.52
CAS Number:
[2548963-55-7]
Formula:
C24H19N7O4S
Target:
Adenosine Receptor|||Carbonic Anhydrase|||Others
T63400
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