GRP78-IN-3, a potent small-molecule-competitive inhibitor of Hsp70 substrate binding and is a selective Grp78 (HSPA5) inhibitor with an IC50 of 0.59 µM. GRP78-IN-3 is 7-fold selective for HspA5 compared to HspA9 (IC50 of 4.3 µM) and >20-fold selective for HspA5 compared to HspA2 (IC50 of 13.9 µM).
Molecular Weight:
342.42
Purity:
99.49%
CAS Number:
[2707510-30-1]
Formula:
C17H18N4O2S
Target:
HSP
T67897
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