WDR5-0102 is a compound that inhibits the WDR5-MLL1 interface (K dis = 7 µM, K d = 4 µM), selectively reducing MLL1 HMT activity without affecting the human H3K4 methyltransferase SETD7 or other HMTs, including G9a, EHMT1, SUV39H2, SETD8, PRMT3, and PRMT5.
Molecular Weight:
374.82
Purity:
98.03%
CAS Number:
[824960-50-1]
Formula:
C18H19ClN4O3
Target:
JAK|||Histone Methyltransferase
T67947
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