GAC0001E5 (1E5) is a dual LXR inverse agonist and degrader (IC50 = 5.4-9.1 µM in pancreatic cancer cells). It inhibits tumor growth and induces apoptosis by promoting LXRalpha/beta degradation and suppressing transcriptional activity.
Molecular Weight:
331.29
Purity:
98.89%
CAS Number:
[927969-67-3]
Formula:
C17H12F3N3O
Target:
Liver X Receptor
T68323
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