Enzastaurin 2HCl, also known as DB-102 and LY317615, is a synthetic macrocyclic bisindolemaleimide with potential antineoplastic activity. Binding to the ATP-binding site, Enzastaurin 2HCl selectively inhibits protein kinase C beta, an enzyme involved in the induction of vascular endothelial growth factor (VEGF)-stimulated neo-angiogenesis. This agent may decrease tumor blood supply and so tumor burden.
Molecular Weight:
588.53
CAS Number:
[365253-37-8]
Formula:
C32H31Cl2N5O2
Target:
Autophagy|||Apoptosis|||Others|||PKC
T69354
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