Relutrigine (PRAX-562) is an orally active, long-acting sodium current inhibitor that preferentially suppresses sustained INa induced by TX-II or SCN8A N1768D mutations (IC50=141/75 nM). It reduces neuronal intrinsic excitability and may be used for anticonvulsant therapy.
Molecular Weight:
407.27
Purity:
99.68%
CAS Number:
[2392951-29-8]
Formula:
C15H11F6N5O2
Target:
Sodium Channel
T69652
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