GSK2807 is a potent and selective, SAM-competitive inhibitor of SMYD3 (Ki = 14 nM). GSK2807 bridges the gap between the SAM-binding pocket and the substrate lysine tunnel of SMYD3. GSK2807 may be useful for cancer treatment.
Molecular Weight:
452.51
CAS Number:
[2245255-65-4]
Formula:
C19H32N8O5
Target:
Histone Methyltransferase|||Others
T69738
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